• Activation and Regioselectivity of Five-Membered Cyclic Thionocarbamates to Nucleophilic Attack 

      Awheda, Ismail; Saygili, Nezire; Garner, A. Christopher; Wallis, John D. (Royal Soc Chemistry, 2013)
      The cyclic thionocarbamate of alaninol undergoes nucleophilic attack by sulfur nucleophiles at 5-C to give 1-thiopropyl-2-amine derivatives when derivatised on nitrogen with a Boc group. Iodide under microwave conditions ...
    • Curcumin-Based Pyrazoline Analogues As Selective Inhibitors Of Human Monoamine Oxidase A 

      Nath, Chandrani; Badavath, Vishnu Nayak; Thakur, Abhishek; Ucar, Gulberk; Acevedo, Orlando; Siddique, Mohd Usman Mohd; Jayaprakash, Venkatesan (Royal Soc Chemistry, 2018)
      A series of 2-methoxy-4-(5-phenyl-4,5-dihydro-1H-pyrazol-3-yl)phenol (pyrazoline) derivatives (2-6) have been synthesized and tested for human monoamine oxidase (hMAO) inhibitory activity. The most active derivative (2) ...